1138245-21-2 Mirogabalin Besylate

Properties

Appearance White to off-white Solid
storage temp. Store at -20°C
solubility DMSO : 125 mg/mL (340.17 mM)
 

Application:

Merogabalin benzenesulfonate is a third-generation calcium channel regulator. Based on the comparative results of various analgesic drugs at home and abroad, targeted optimization has been carried out. Merogabalin has a strong binding affinity for the α 2 δ -1 subunit, slow dissociation from the α 2 δ -1 subunit, and rapid dissociation from the α 2 δ -2 subunit. This may be the reason why Merogabalin has better analgesic treatment effect and fewer adverse reactions. In preclinical studies, its analgesic effect is stronger and more lasting than pregabalin

 

Synonyms:

Mirogabalin besylate

1138245-21-2

2-[(1R,5S,6S)-6-(aminomethyl)-3-ethyl-6-bicyclo[3.2.0]hept-3-enyl]acetic acid;benzenesulfonic acid

Mirogabalin besilate 

Bicyclo(3.2.0)hept-3-ene-6-acetic acid, 6-(aminomethyl)-3-ethyl-, (1R,5S,6S)-, benzenesulfonate (1:1)

2-((1R,5S,6S)-6-(aminomethyl)-3-ethylbicyclo[3.2.0]hept-3-en-6-yl)acetic acid compound with benzenesulfonic acid (1:1)

benzenesulfonic acid; mirogabalin

2-((1R,5S,6S)-6-(aminomethyl)-3-ethylbicyclo[3.2.0]hept-3-en-6-yl)acetic acid besylate

Mirogabalin besylate

C18H25NO5S

2-[(1R,5S,6S)-6-(aminomethyl)-3-ethylbicyclo[3.2.0]hept-3-en-6-yl]acetic acid; benzenesulfonic acid

EX-A2817

2-((1R,5S,6S)-6-(aminomethyl)-3-ethylbicyclo[3.2.0]hept-3-en-6-yl)aceticacidbesylate

[(1R,5S,6S)-6-(Aminomethyl)-3-ethylbicyclo[3.2.0]hept-3-en-6-yl]acetic acid monobenzenesulfonate

 

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