832720-36-2 Elagolix Sodium

Properties

Appearance White to Off-White Solid
Melting point:>188°C (dec.)
storage temp. Hygroscopic, -20°C Freezer, Under inert atmosphere
solubility DMSO (Slightly), Methanol (Slightly)
Water Solubility H2O: 2mg/mL, clear
Stability:Hygroscopic

 

Application:

Elagolix sodium is a human GnRH receptor (GnRHR) antagonist with an IC50 of 0.25 nM in kinase assays [1].
It also showed NFAT inhibition with an IC50 of 5.4 nM and effectively blocked Ca2+flux with an IC50 of 0.86 nM [1].

 

Synonyms:

Elagolix sodium

832720-36-2

Elagolix sodium salt

Orlissa

5948VUI423

832720-36-2 (sodium)

sodium (R)-4-((2-(5-(2-fluoro-3-methoxyphenyl)-3-(2-fluoro-6-(trifluoromethyl)benzyl)-4-methyl-2,6-dioxo-2,3-dihydropyrimidin-1(6H)-yl)-1-phenylethyl)amino)butanoate

ORIAHNN COMPONENT ELAGOLIX SODIUM

Elagolix sodium

sodium;4-[[(1R)-2-[5-(2-fluoro-3-methoxyphenyl)-3-[[2-fluoro-6-(trifluoromethyl)phenyl]methyl]-4-methyl-2,6-dioxopyrimidin-1-yl]-1-phenylethyl]amino]butanoate

CHEMBL502182

Butanoic acid, 4-(((1R)-2-(5-(2-fluoro-3-methoxyphenyl)-3-((2-fluoro-6-(trifluoromethyl)phenyl)methyl)-3,6-dihydro-4-methyl-2,6-dioxo-1(2H)-pyrimidinyl)-1-phenylethyl)amino)-, monosodium salt

Sodium 4-(((1R)-2-(5-(2-fluoro-3-methoxyphenyl)-3-((2-fluoro-6-(trifluoromethyl)phenyl)methyl)-4-methyl-2,6-dioxo-3,6-dihydropyrimidin-1(2H)-yl)-1-phenylethyl)amino)butanoate

Elagolix sodium

Orilissa 

NBI-56418 sodium

Elagolix sodium (Standard)

DTXSID601003247

GLXC-10785

ELAGOLIX SODIUM [ORANGE BOOK]

ELAGOLIX SODIUM COMPONENT OF ORIAHNN

4-((r)-2-[5-(2-fluoro-3-methoxy-phenyl)-3-(2-fluoro-6-trifluoromethyl-benzyl)-4-methyl-2,6-dioxo-3,6-dihydro-2h-pyrimidin-1-yl]-1-phenyl-ethylamino)-butyric acid sodium salt

 

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